Enalapril Maleate
Latar mburi
Enalapril Maleate
Katrangan
Enalapril (maleate) (MK-421 (maleate)), metabolit aktif enalapril, minangka inhibitor enzim konversi angiotensin (ACE).
Ing Vivo
Enalapril (MK-421) minangka prodrug sing kalebu kelas obat-obatan inhibitor angiotensin-converting enzyme (ACE).Metabolisme kanthi cepet ing ati dadi enalaprilat sawise administrasi oral.Enalapril (MK-421) minangka inhibitor kompetitif ACE sing kuat, enzim sing tanggung jawab kanggo konversi angiotensin I (ATI) dadi angiotensin II (ATII).ATII ngatur tekanan getih lan minangka komponen kunci saka sistem renin-angiotensin-aldosteron (RAAS).Enalapril bisa digunakake kanggo nambani hipertensi esensial utawa renovaskular lan gagal jantung kongestif gejala.
Lumbung
bubuk | -20°C | 3 taun |
4°C | 2 taun | |
Ing solvent | -80°C | 6 wulan |
-20°C | 1 wulan |
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